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Information × Registration Number 0217U001887, 0114U001342 , R & D reports Title The search for new potential biologicallyactive substances in a series of fused-imidazole and its heteroanalogue popup.stage_title Head Demchenko Anatolij Michajlovich Bukhtiarova Tatiana Anatoliivna, Registration Date 02-08-2017 Organization State Establishment "Institute of Pharmacology and Toxicology National Academy of Medical Science of Ukraine" popup.description2 Developed methods of synthesis of 98 new fused imidazole compounds (imidazothiazines, imidazoazepines, imidazopyridines) and imidazole heteroanalogues (pyrrolopyridines, triazoloazepines, triazacyclopent [cd]azulenes, triazolopyrimidines, triazolothiadiazines, thiazolopyridazinones). Performed screening in silico, in vivo of the target biological activity species - analgesic, anti-inflammatory and anti-tumor. Obtained compounds leaders, promising to study in depth. Product Description popup.authors Бобкова Л.С. Голубов М.І. Демченко С.А. Дудник А.Є. Козлик В.В. Мєшкова Н. Максюта С.В. Омельяненко З.П. Сергеєв В.С. Серединська Н.М. Татьянченко І.С. Хавич О.О. Хайрулін А.Р. Хоменко В.С. Шарикіна Н.І. popup.nrat_date 2020-04-02 Close